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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T28482 |
Firibastat
QGC 001,QGC-001,RB-150,RB150,QGC001,RB 150 |
Aminopeptidase | Metabolism |
Firibastat (RB150) 是一种具有口服活性的 EC33 前体药物。Firibastat 是一种首创的脑氨基肽酶 A(APA) 抑制剂 (Ki=200 nM),选择性地抑制高血压大鼠脑血管紧张素 II 转化为血管紧张素 III,降低血压。 | |||
T36943 | Aminopeptidase N Inhibitor | ||
Aminopeptidase N (AP-N) inhibitor is a reversible inhibitor of AP-N/CD13 (IC50 = 25 μM). It is selective for AP-N/CD13 over matrix metalloproteinase-9 (MMP-9), angiotensin converting enzyme (ACE), neutral endopeptidase (NEP), γ-glutamyl transpeptidase, and the serine proteases dipeptidyl peptidase 4 (DPP-4) and cathepsin G at a concentration of 1 mM. AP-N inhibitor is non-cytotoxic to U937 cells at a concentration of 100 μM. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T11203 |
Enocyanin
|
Others | Others |
Enocyanin, an anthocyanin extracted from grapes, exhibits inhibitory effects on leucine aminopeptidase, acid phosphatase, γ-glutamyl transpeptidase, and esterase activity. |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-03041 |
Aminopeptidase A Protein, Rat, Recombinant (aa 41-945, His)
ENPEP,glutamyl aminopeptidase |
Rat | Baculovirus Insect Cells |
Aminopeptidase A Protein, Rat, Recombinant (aa 41-945, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 106 kDa and the accession number is P50123-1. | |||
TMPY-00644 |
Aminopeptidase A Protein, Human, Recombinant (His)
APA,glutamyl aminopeptidase,ENPEP,gp160,CD... |
Human | Baculovirus Insect Cells |
Aminopeptidase A Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 107.2 kDa and the accession number is Q07075. | |||
TMPY-02896 |
Aminopeptidase A Protein, Mouse, Recombinant (His)
Ly-51,6030431M22Rik,ENPEP,APA,Bp-1/6C3,glutamyl |
Mouse | Baculovirus Insect Cells |
Aminopeptidase A Protein, Mouse, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 106 kDa and the accession number is P16406. |